| 論文 |
papers |
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High-throughput phenotypic screening identifies novel antimalarial scaffolds and target-associated chemotypes Japheth Kibet Ng’etich,Normalita Eka Pravitasari,Takeshi Ishikawa,Naoya Kadofusa,Ayato Sato,Shinjiro Hamano,Takaya Sakura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 100658頁-100658頁 2026年07月
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Antiviral activities of ascofuranone and naphthoquinone derivatives against Ebola virus Christelle M. Pemba,Yasuteru Sakurai,Yohei Kurosaki,J.J. Patten,Eri Amalia,Daniel K. Inaoka,Robert A. Davey,Tomoo Shiba,Kiyoshi Kita,Jiro Yasuda Antiviral Research 249巻106400頁-106400頁 2026年05月
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Crystallographic snapshots of Trypanosoma cruzi aspartate transcarbamoylase including catalytic intermediates suggest an ordered Bi–Bi reaction mechanism Kazuaki Matoba,Takeshi Nara,Takashi Aoki,Teruki Honma,Akiko Tanaka,Masayuki Inoue,Shigeru Matsuoka,Shigeharu Harada,Kiyoshi Kita,Daniel Ken Inaoka,Emmanuel Oluwadare Balogun,Tomoo Shiba Scientific Reports 2026年04月02日
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A novel 2-piperazino-pyrimidine compound exhibits asexual antimalarial activity by targeting Plasmodium falciparum plasmepsin X Jing Hong,Takaya Sakura,Naoya Asada,Kouki Fuchino,Daiki Kuwana,Rina Kaki,Ryuta Ishii,Teruhisa Kato,Kiyoshi Kita,Kenichi Matsumura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 100644頁-100644頁 2026年04月
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Distinct quaternary reaction behavior and stable charge-transfer complex formation in Schistosoma mansoni sulfide:quinone oxidoreductase Augustin Tshibaka Kabongo,Talaam Keith Kiplangat,Yuki Tayama,Acharjee Rajib,Yuichi Matsuo,Linh Manh Ha,Samandram Sushilkumar Singh,Tetsuo Yamashita,Euki Yazaki,Endah Dwi Hartuti,Tetsuro Matsunaga,Tomoaki Ida,Tomoyoshi Nozaki,Takaaki Akaike,Tomoo Shiba,Jun-ichi Kishikawa,Shinjiro Hamano,Kiyoshi Kita,Daniel Ken Inaoka Free Radical Biology and Medicine 2026年02月
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Modulation of succinyl‐CoA:3‐ketoacid CoA transferase activity by a single amino acid residue in acetate:succinate CoA transferase from Trypanosoma brucei, the causative agent of African sleeping sickness Kota Mochizuki,Daniel Ken Inaoka,Keisuke Fukuda,Hana Kurasawa,Kenji Iyoda,Uta Nakai,Shigeharu Harada,Emmanuel O. Balogun,Frédéric Bringaud,Michael Boshart,Takaya Sakura,Kenji Hirayama,Kiyoshi Kita,Tomoo Shiba Protein Science 35巻2号 2026年01月20日
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Plasmodium falciparum diacylglycerol acyltransferase maintains phospholipid homeostasis to regulate sexual differentiation, ER stress, and cytoadhesion Minako Yoshida,Junpei Fukumoto,Shinya Miyazaki,Megumi Tanaka,Suzumi M Tokuoka,Hideru Obinata,Takaya Sakura,Yoko Onizuka,Daniel Ken Inaoka,Kiyoshi Kita,Kazuhide Yahata,Eizo Takashima,Hideo Shindou,Fuyuki Tokumasu 2025年10月13日
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DNA Vaccine Encoding Trypanosoma brucei MSP‐B Elicited IgG and IFN‐γ Responses and Partial Protection in Immunised Mice Aminu Bashir Yusuf,Edwige Flore Gouegni,Amaya Jobin Habila,Isma'ila Alhaji Umar,Sani Ibrahim,Junaid Kabir,Kenji Hirayama,Kentaro Kato,Clara Vasquez Velasquez,Daniel Ken Inaoka,Mohammed Mamman,Emmanuel Oluwadare Balogun,Mohammed Nasir Shuaibu Parasite Immunology 47巻10号 2025年10月09日
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The Extracellular Region of Trypanosoma congolense Membrane Bound Acid Phosphatase Induces Partial Protection in Immunized BALB/c mice Gouegni E. Flore,Aminu B. Yusuf,Amaya J. Habila,Mohammed Mamman,Sunday E. Atawodi,Kentaro Kato,Daniel K. Inaoka,Kenji Hirayama,Kiyoshi Kita,Mohammed N. Shuaibu,Emmanuel O. Balogun Microbial Pathogenesis 107526頁-107526頁 2025年04月
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Development of tolerance to bedaquiline by overexpression of trypanosomal acetate: succinate CoA transferase in Mycobacterium smegmatis Bundutidi GM,Mochizuki K.,Matsuo Y.,Hayashishita M.,Sakura T.,Ando Y.,Cook GM,Rajib A.,Bringaud F.,Boshart M.,Hamano S.,Sekijima M.,Hirayama K.,Kita K.,Inaoka DK Commmunications Biology 8巻1号187頁- 2025年02月
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High-throughput phenotypic screening identifies novel antimalarial scaffolds and target-associated chemotypes Japheth Kibet Ng’etich,Normalita Eka Pravitasari,Takeshi Ishikawa,Naoya Kadofusa,Ayato Sato,Shinjiro Hamano,Takaya Sakura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 100658-100658 2026/07
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Antiviral activities of ascofuranone and naphthoquinone derivatives against Ebola virus Christelle M. Pemba,Yasuteru Sakurai,Yohei Kurosaki,J.J. Patten,Eri Amalia,Daniel K. Inaoka,Robert A. Davey,Tomoo Shiba,Kiyoshi Kita,Jiro Yasuda Antiviral Research 249.106400-106400 2026/05
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Crystallographic snapshots of Trypanosoma cruzi aspartate transcarbamoylase including catalytic intermediates suggest an ordered Bi–Bi reaction mechanism Kazuaki Matoba,Takeshi Nara,Takashi Aoki,Teruki Honma,Akiko Tanaka,Masayuki Inoue,Shigeru Matsuoka,Shigeharu Harada,Kiyoshi Kita,Daniel Ken Inaoka,Emmanuel Oluwadare Balogun,Tomoo Shiba Scientific Reports 2026/04/02
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A novel 2-piperazino-pyrimidine compound exhibits asexual antimalarial activity by targeting Plasmodium falciparum plasmepsin X Jing Hong,Takaya Sakura,Naoya Asada,Kouki Fuchino,Daiki Kuwana,Rina Kaki,Ryuta Ishii,Teruhisa Kato,Kiyoshi Kita,Kenichi Matsumura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 100644-100644 2026/04
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Distinct quaternary reaction behavior and stable charge-transfer complex formation in Schistosoma mansoni sulfide:quinone oxidoreductase Augustin Tshibaka Kabongo,Talaam Keith Kiplangat,Yuki Tayama,Acharjee Rajib,Yuichi Matsuo,Linh Manh Ha,Samandram Sushilkumar Singh,Tetsuo Yamashita,Euki Yazaki,Endah Dwi Hartuti,Tetsuro Matsunaga,Tomoaki Ida,Tomoyoshi Nozaki,Takaaki Akaike,Tomoo Shiba,Jun-ichi Kishikawa,Shinjiro Hamano,Kiyoshi Kita,Daniel Ken Inaoka Free Radical Biology and Medicine 2026/02
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Modulation of succinyl‐CoA:3‐ketoacid CoA transferase activity by a single amino acid residue in acetate:succinate CoA transferase from Trypanosoma brucei, the causative agent of African sleeping sickness Kota Mochizuki,Daniel Ken Inaoka,Keisuke Fukuda,Hana Kurasawa,Kenji Iyoda,Uta Nakai,Shigeharu Harada,Emmanuel O. Balogun,Frédéric Bringaud,Michael Boshart,Takaya Sakura,Kenji Hirayama,Kiyoshi Kita,Tomoo Shiba Protein Science 35.2. 2026/01/20
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Plasmodium falciparum diacylglycerol acyltransferase maintains phospholipid homeostasis to regulate sexual differentiation, ER stress, and cytoadhesion Minako Yoshida,Junpei Fukumoto,Shinya Miyazaki,Megumi Tanaka,Suzumi M Tokuoka,Hideru Obinata,Takaya Sakura,Yoko Onizuka,Daniel Ken Inaoka,Kiyoshi Kita,Kazuhide Yahata,Eizo Takashima,Hideo Shindou,Fuyuki Tokumasu 2025/10/13
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DNA Vaccine Encoding Trypanosoma brucei MSP‐B Elicited IgG and IFN‐γ Responses and Partial Protection in Immunised Mice Aminu Bashir Yusuf,Edwige Flore Gouegni,Amaya Jobin Habila,Isma'ila Alhaji Umar,Sani Ibrahim,Junaid Kabir,Kenji Hirayama,Kentaro Kato,Clara Vasquez Velasquez,Daniel Ken Inaoka,Mohammed Mamman,Emmanuel Oluwadare Balogun,Mohammed Nasir Shuaibu Parasite Immunology 47.10. 2025/10/09
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The Extracellular Region of Trypanosoma congolense Membrane Bound Acid Phosphatase Induces Partial Protection in Immunized BALB/c mice Gouegni E. Flore,Aminu B. Yusuf,Amaya J. Habila,Mohammed Mamman,Sunday E. Atawodi,Kentaro Kato,Daniel K. Inaoka,Kenji Hirayama,Kiyoshi Kita,Mohammed N. Shuaibu,Emmanuel O. Balogun Microbial Pathogenesis 107526-107526 2025/04
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Development of tolerance to bedaquiline by overexpression of trypanosomal acetate: succinate CoA transferase in Mycobacterium smegmatis Bundutidi GM,Mochizuki K.,Matsuo Y.,Hayashishita M.,Sakura T.,Ando Y.,Cook GM,Rajib A.,Bringaud F.,Boshart M.,Hamano S.,Sekijima M.,Hirayama K.,Kita K.,Inaoka DK Commmunications Biology 8.1.187- 2025/02
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