| 論文 |
papers |
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A novel 2-piperazino-pyrimidine compound exhibits asexual antimalarial activity by targeting Plasmodium falciparum plasmepsin X Jing Hong,Takaya Sakura,Naoya Asada,Kouki Fuchino,Daiki Kuwana,Rina Kaki,Ryuta Ishii,Teruhisa Kato,Kiyoshi Kita,Kenichi Matsumura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 31巻100644頁-100644頁 2026年08月
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High-throughput phenotypic screening identifies novel antimalarial scaffolds and target-associated chemotypes Japheth Kibet Ng'etich,Normalita Eka Pravitasari,Takeshi Ishikawa,Naoya Kadofusa,Ayato Sato,Shinjiro Hamano,Takaya Sakura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 31巻100658頁-100658頁 2026年08月
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Epigenetic landscape of the H3K27me3 mark in macrophages transformed by Theileria annulata Takaya Sakura,Shahin Tajeri,Zineb Rchiad,Hifzur R. Ansari,Abhinav Kaushik,Tobias Mourier,Arnab Pain,Michel Wassef,Gordon Langsley Communications Biology 2026年02月24日
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Modulation of succinyl-CoA:3-ketoacid CoA transferase activity by a single amino acid residue in acetate:succinate CoA transferase from Trypanosoma brucei, the causative agent of African sleeping sickness Kota Mochizuki,Daniel Ken Inaoka,Keisuke Fukuda,Hana Kurasawa,Kenji Iyoda,Uta Nakai,Shigeharu Harada,Emmanuel O. Balogun,Frédéric Bringaud,Michael Boshart,Takaya Sakura,Kenji Hirayama,Kiyoshi Kita,Tomoo Shiba Protein Science 35巻2号 2026年01月20日
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Plasmodium falciparum diacylglycerol acyltransferase maintains phospholipid homeostasis to regulate sexual differentiation, ER stress, and cytoadhesion Minako Yoshida,Junpei Fukumoto,Shinya Miyazaki,Megumi Tanaka,Suzumi M Tokuoka,Hideru Obinata,Takaya Sakura,Yoko Onizuka,Daniel Ken Inaoka,Kiyoshi Kita,Kazuhide Yahata,Eizo Takashima,Hideo Shindou,Fuyuki Tokumasu 2025年10月13日
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Development of tolerance to bedaquiline by overexpression of trypanosomal acetate: succinate CoA transferase in Mycobacterium smegmatis Gloria Mavinga Bundutidi,Kota Mochizuki,Yuichi Matsuo,Mizuki Hayashishita,Takaya Sakura,Yuri Ando,Gregory Murray Cook,Acharjee Rajib,Frédéric Bringaud,Michael Boshart,Shinjiro Hamano,Masakazu Sekijima,Kenji Hirayama,Kiyoshi Kita,Daniel Ken Inaoka Communications Biology 8巻1号 2025年02月06日
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Pivotal roles of Plasmodium falciparum lysophospholipid acyltransferase 1 in cell cycle progression and cytostome internalization Junpei Fukumoto,Minako Yoshida,Suzumi M. Tokuoka,Eri Saki H. Hayakawa,Shinya Miyazaki,Takaya Sakura,Daniel Ken Inaoka,Kiyoshi Kita,Jiro Usukura,Hideo Shindou,Fuyuki Tokumasu Communications Biology 8巻1号 2025年01月29日
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Accelerating antimalarial drug discovery with a new high-throughput screen for fast-killing compounds Takaya Sakura,Ryuta Ishii,Eri Yoshida,Kiyoshi Kita,Teruhisa Kato,Daniel Ken Inaoka ACS Infectious Diseases 2024年11月19日
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Glycolytic enzymes form membrane-less condensates in the malaria parasite Plasmodium falciparum by sensing glucose levels Ryuta Ishii,Takaya Sakura,Daniel Ken Inaoka,Fuyuki Tokumasu 2024年04月11日
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Effect of geranylated dihydrochalcone from Artocarpus altilis leaves extract on Plasmodium falciparum ultrastructural changes and mitochondrial malate: Quinone oxidoreductase Agriana Rosmalina Hidayati,Melinda,Hilkatul Ilmi,Takaya Sakura,Miako Sakaguchi,Junko Ohmori,Endah Dwi Hartuti,Lidya Tumewu,Daniel Ken Inaoka,Mulyadi Tanjung,Eri Yoshida,Fuyuki Tokumasu,Kiyoshi Kita,Mihoko Mori,Kazuyuki Dobashi,Tomoyoshi Nozaki,Din Syafruddin,Achmad Fuad Hafid,Danang Waluyo,Aty Widyawaruyanti International Journal for Parasitology: Drugs and Drug Resistance 21巻40頁-50頁 2023年04月
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A novel 2-piperazino-pyrimidine compound exhibits asexual antimalarial activity by targeting Plasmodium falciparum plasmepsin X Jing Hong,Takaya Sakura,Naoya Asada,Kouki Fuchino,Daiki Kuwana,Rina Kaki,Ryuta Ishii,Teruhisa Kato,Kiyoshi Kita,Kenichi Matsumura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 31.100644-100644 2026/08
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High-throughput phenotypic screening identifies novel antimalarial scaffolds and target-associated chemotypes Japheth Kibet Ng'etich,Normalita Eka Pravitasari,Takeshi Ishikawa,Naoya Kadofusa,Ayato Sato,Shinjiro Hamano,Takaya Sakura,Daniel Ken Inaoka International Journal for Parasitology: Drugs and Drug Resistance 31.100658-100658 2026/08
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Epigenetic landscape of the H3K27me3 mark in macrophages transformed by Theileria annulata Takaya Sakura,Shahin Tajeri,Zineb Rchiad,Hifzur R. Ansari,Abhinav Kaushik,Tobias Mourier,Arnab Pain,Michel Wassef,Gordon Langsley Communications Biology 2026/02/24
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Modulation of succinyl-CoA:3-ketoacid CoA transferase activity by a single amino acid residue in acetate:succinate CoA transferase from Trypanosoma brucei, the causative agent of African sleeping sickness Kota Mochizuki,Daniel Ken Inaoka,Keisuke Fukuda,Hana Kurasawa,Kenji Iyoda,Uta Nakai,Shigeharu Harada,Emmanuel O. Balogun,Frédéric Bringaud,Michael Boshart,Takaya Sakura,Kenji Hirayama,Kiyoshi Kita,Tomoo Shiba Protein Science 35.2. 2026/01/20
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Plasmodium falciparum diacylglycerol acyltransferase maintains phospholipid homeostasis to regulate sexual differentiation, ER stress, and cytoadhesion Minako Yoshida,Junpei Fukumoto,Shinya Miyazaki,Megumi Tanaka,Suzumi M Tokuoka,Hideru Obinata,Takaya Sakura,Yoko Onizuka,Daniel Ken Inaoka,Kiyoshi Kita,Kazuhide Yahata,Eizo Takashima,Hideo Shindou,Fuyuki Tokumasu 2025/10/13
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Development of tolerance to bedaquiline by overexpression of trypanosomal acetate: succinate CoA transferase in Mycobacterium smegmatis Gloria Mavinga Bundutidi,Kota Mochizuki,Yuichi Matsuo,Mizuki Hayashishita,Takaya Sakura,Yuri Ando,Gregory Murray Cook,Acharjee Rajib,Frédéric Bringaud,Michael Boshart,Shinjiro Hamano,Masakazu Sekijima,Kenji Hirayama,Kiyoshi Kita,Daniel Ken Inaoka Communications Biology 8.1. 2025/02/06
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Pivotal roles of Plasmodium falciparum lysophospholipid acyltransferase 1 in cell cycle progression and cytostome internalization Junpei Fukumoto,Minako Yoshida,Suzumi M. Tokuoka,Eri Saki H. Hayakawa,Shinya Miyazaki,Takaya Sakura,Daniel Ken Inaoka,Kiyoshi Kita,Jiro Usukura,Hideo Shindou,Fuyuki Tokumasu Communications Biology 8.1. 2025/01/29
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Accelerating antimalarial drug discovery with a new high-throughput screen for fast-killing compounds Takaya Sakura,Ryuta Ishii,Eri Yoshida,Kiyoshi Kita,Teruhisa Kato,Daniel Ken Inaoka ACS Infectious Diseases 2024/11/19
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Glycolytic enzymes form membrane-less condensates in the malaria parasite Plasmodium falciparum by sensing glucose levels Ryuta Ishii,Takaya Sakura,Daniel Ken Inaoka,Fuyuki Tokumasu 2024/04/11
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Effect of geranylated dihydrochalcone from Artocarpus altilis leaves extract on Plasmodium falciparum ultrastructural changes and mitochondrial malate: Quinone oxidoreductase Agriana Rosmalina Hidayati,Melinda,Hilkatul Ilmi,Takaya Sakura,Miako Sakaguchi,Junko Ohmori,Endah Dwi Hartuti,Lidya Tumewu,Daniel Ken Inaoka,Mulyadi Tanjung,Eri Yoshida,Fuyuki Tokumasu,Kiyoshi Kita,Mihoko Mori,Kazuyuki Dobashi,Tomoyoshi Nozaki,Din Syafruddin,Achmad Fuad Hafid,Danang Waluyo,Aty Widyawaruyanti International Journal for Parasitology: Drugs and Drug Resistance 21.40-50 2023/04
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